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Isoform of the progesterone receptor
The progesterone receptor C (PR-C) is one of three known
isoforms of the
progesterone receptor (PR), the main
biological target of the
endogenous
progestogen
sex hormone
progesterone.
[1]
[2] The other isoforms of the PR include the
PR-A and
PR-B.
[1]
[2]
See also
References
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(1) Basic domains |
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(1.1) Basic
leucine zipper (
bZIP) | |
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(1.2) Basic helix-loop-helix (
bHLH) | Group A | |
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Group B | |
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Group C bHLH-
PAS | |
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Group D | |
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Group E | |
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Group F bHLH-COE | |
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(1.3)
bHLH-ZIP | |
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(1.4) NF-1 | |
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(1.5) RF-X | |
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(1.6) Basic helix-span-helix (bHSH) | |
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(2)
Zinc finger DNA-binding domains |
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(2.1)
Nuclear receptor (Cys4) | subfamily 1 | |
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subfamily 2 | |
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subfamily 3 | |
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subfamily 4 | |
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subfamily 5 | |
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subfamily 6 | |
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subfamily 0 | |
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(2.2) Other Cys4 | |
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(2.3) Cys2His2 | |
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(2.4) Cys6 | |
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(2.5) Alternating composition | |
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(2.6) WRKY | |
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(4) β-Scaffold factors with minor groove contacts |
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(0) Other transcription factors |
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PRTooltip Progesterone receptor | Agonists |
- Testosterone derivatives: Progestins:
6,6-Difluoronorethisterone
-
6,6-Difluoronorethisterone acetate
-
17α-Allyl-19-nortestosterone
-
Allylestrenol
-
Altrenogest
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Chloroethynylnorgestrel
-
Cingestol
-
Danazol
-
Desogestrel
-
Dienogest
-
Ethinylandrostenediol
-
Ethisterone
-
Ethynerone
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Etonogestrel
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Etynodiol
-
Etynodiol diacetate
-
Gestodene
-
Gestrinone
-
Levonorgestrel
-
Levonorgestrel esters (e.g.,
levonorgestrel butanoate)
-
Lynestrenol
-
Lynestrenol phenylpropionate
-
Metynodiol
-
Metynodiol diacetate
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Norelgestromin
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Norethisterone (norethindrone)
-
Norethisterone esters (e.g.,
norethisterone acetate,
norethisterone enanthate)
-
Noretynodrel
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Norgesterone
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Norgestimate
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Norgestrel
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Norgestrienone
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Norvinisterone
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Oxendolone
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Quingestanol
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Quingestanol acetate
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Tibolone
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Tigestol
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Tosagestin; Anabolic–androgenic steroids:
11β-Methyl-19-nortestosterone
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11β-Methyl-19-nortestosterone dodecylcarbonate
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19-Nor-5-androstenediol
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19-Nor-5-androstenedione
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19-Nordehydroepiandrosterone
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Bolandiol
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Bolandiol dipropionate
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Bolandione
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Dimethisterone
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Dienedione
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Dienolone
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Dimethandrolone
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Dimethandrolone buciclate
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Dimethandrolone dodecylcarbonate
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Dimethandrolone undecanoate
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Dimethyldienolone
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Dimethyltrienolone
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Ethyldienolone
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Ethylestrenol (ethylnandrol)
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Methyldienolone
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Metribolone (R-1881)
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Methoxydienone (methoxygonadiene)
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Mibolerone
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Nandrolone
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Nandrolone esters (e.g.,
nandrolone decanoate,
nandrolone phenylpropionate)
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Norethandrolone
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Normethandrone (methylestrenolone, normethandrolone, normethisterone)
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RU-2309
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Tetrahydrogestrinone
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Trenbolone (trienolone)
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Trenbolone esters (e.g.,
trenbolone acetate,
trenbolone enanthate)
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Trendione
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Trestolone
-
Trestolone acetate
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Mixed (
SPRMsTooltip Selective progesterone receptor modulators) | |
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Antagonists | |
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mPRTooltip Membrane progesterone receptor (
PAQRTooltip Progestin and adipoQ receptor) | |
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