From Wikipedia, the free encyclopedia
Chemical compound
Deschloroetizolam
Dependence liability Moderate
Routes of administration Oral, sublingual, rectal
Legal status
DE :
NpSG (Industrial and scientific use only)
UK :
Class C
Illegal in Sweden
4-phenyl-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine
CAS Number
PubChem
CID
ChemSpider
UNII
Formula C 17 H 16 N 4 S
Molar mass 308.40 g·mol−1 3D model (
JSmol )
CCC1=CC2=C(S1)N3C(=NN=C3CN=C2C4=CC=CC=C4)C
InChI=1S/C17H16N4S/c1-3-13-9-14-16(12-7-5-4-6-8-12)18-10-15-20-19-11(2)21(15)17(14)22-13/h4-9H,3,10H2,1-2H3
Key:JIOBORXCOGMHSV-UHFFFAOYSA-N
Deschloroetizolam (also known as Etizolam-2 ) is a
thienotriazolodiazepine that is the dechlorinated
analog of the closely related
etizolam .
[1]
[2]
[3] The compound has been sold as a
designer drug .
[4]
[5]
[6]
[7]
Legal status
Deschloroetizolam is classified and controlled as a hazardous substance in Sweden as of on October 15, 2015.
[8]
See also
References
^ Weber KH, Bauer A, Langbein A, Daniel H (September 1978). "Heteroaromaten mit anellierten Siebenringen, III. Umwandlung von Thienotriazolooxazepinen in Diazepine". Justus Liebigs Annalen der Chemie (in German). 1978 (8): 1257–1265.
doi :
10.1002/jlac.197819780806 .
^
US 3904641 , Nakanishi M, Tahara T, Araki K, Shiroki M, "Triazolothienodiazepine compounds", published 1975-09-09, assigned to Yoshitomi Pharmaceutical Industries, Ltd.
^
EP 0776892 , Hiroshi K, Syuji E, Hideaki S, Minoru M, Kenichi O, "Thienylazole compound and thienotriazolodiazepine compound", published 4 June 1997, assigned to Yoshitomi Pharmaceutical Industries, Ltd.
^
"Deschloroetizolam" . New Synthetic Drugs Database. 9 November 2023.
^ Pettersson Bergstrand M, Helander A, Hansson T, Beck O (April 2017). "Detectability of designer benzodiazepines in CEDIA, EMIT II Plus, HEIA, and KIMS II immunochemical screening assays". Drug Testing and Analysis . 9 (4): 640–645.
doi :
10.1002/dta.2003 .
PMID
27366870 .
^ Manchester KR, Maskell PD, Waters L (March 2018).
"Experimental versus theoretical log D7.4 , pKa and plasma protein binding values for benzodiazepines appearing as new psychoactive substances" . Drug Testing and Analysis . 10 (8): 1258–1269.
doi :
10.1002/dta.2387 .
PMID
29582576 .
S2CID
31098917 .
^ Manchester KR, Waters L, Haider S, Maskell PD (July 2022).
"The blood-to-plasma ratio and predicted GABAA -binding affinity of designer benzodiazepines" . Forensic Toxicology . 40 (2): 349–356.
doi :
10.1007/s11419-022-00616-y .
PMC
9715504 .
PMID
36454409 .
S2CID
247455284 .
^
"Nya substanser klassas som narkotika eller hälsofarlig vara" (in Swedish). Folkhälsomyndigheten. 18 August 2015.
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